SCHEMBL8780428

SCHEMBL8780428

CCc1nc2c(C(F)(F)F)cccc2c(O)c1C(=O)OC(C)CC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
LMNA P02545 2/20 0.38
GLA P06280 2/20 0.38
GAA P10253 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
GABRA1 P14867 3/20 0.38
GABRG2 P18507 3/20 0.38
GABRB3 P28472 3/20 0.38
GABRA5 P31644 3/20 0.38
GABRA3 P34903 3/20 0.38
GABRA2 P47869 3/20 0.38
GABRA6 Q16445 1/20 0.38
MAPT P10636 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10946606 0.84 KDM4E (0.46) ALDH1A1KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL11043805 0.81 P2RX3 (0.41) NR1H2NR1H3KCNH2
SCHEMBL11623025 0.78 KDM4E (0.43) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL8780458 0.78 USP2 (0.47) HSD17B10GABRA1GABRG2GABRB3GABRA5
SCHEMBL11622215 0.76 ALOX5 (0.46) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL10946317 0.76 KDM4E (0.52) ALDH1A1KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL11617193 0.76 KDM4E (0.44) ALDH1A1KDM4ELMNAHSD17B10MAPT
SCHEMBL8780497 0.74 APLNR (0.44) ALDH1A1KDM4ELMNAHSD17B10MAPT
SCHEMBL11615579 0.74 P2RX3 (0.41) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL11619432 0.73 KDM4E (0.44) ALDH1A1KDM4EHPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP claimed