SCHEMBL8780434

SCHEMBL8780434

CN(C)Cc1ccc(C2(O)CCC(=O)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.41
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
OPRM1 P35372 3/20 0.37
OPRK1 P41145 3/20 0.37
OPRL1 P41146 3/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LSS P48449 1/20 0.35
OPRD1 P41143 1/20 0.34
PARP1 P09874 3/20 0.33
GRM2 Q14416 1/20 0.33
BRD4 O60885 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
TTK P33981 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethylene SCHEMBL8389434 0.97 HRH3 (0.39) HRH3ALDH1A1TSHRTAAR1OPRM1
SCHEMBL11800411 0.81 OPRL1 (0.49) ALDH1A1OPRM1OPRK1OPRL1OPRD1
SCHEMBL613533 0.78 OPRL1 (0.49) ALDH1A1TSHROPRM1OPRK1OPRL1
SCHEMBL745497 0.78 CHRNB2 (0.34) HRH3PARP1CHEK1MAP2K1
SCHEMBL27611842 0.76 HRH3 (0.43) HRH3ALDH1A1TSHROPRM1OPRK1
SCHEMBL613284 0.75 OPRM1 (0.49) OPRM1OPRK1OPRL1OPRD1PARP1
SCHEMBL8534738 0.75 SLC6A4 (0.44) HRH3ALDH1A1TSHRTAAR1OPRM1
SCHEMBL612855 0.73 ESR2 (0.43) MEN1CYP2C9KMT2A
SCHEMBL613957 0.72 DRD2 (0.58) ALDH1A1TSHROPRM1OPRK1OPRL1
SCHEMBL613615 0.72 OPRM1 (0.45) TSHROPRM1OPRK1OPRL1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757669-A1 O-ACYL-4-PHENYL-CYCLOHEXANOLS, THEIR SALTS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE, AS WELL AS A METHOD OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-02-12 EP disclosed
WO-1995029148-A1 O-ACYL-4-PHENYL-CYCLOHEXANOLS, THEIR SALTS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE, AS WELL AS A METHOD OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1995-11-02 WO disclosed