SCHEMBL8534738

SCHEMBL8534738

CN(C)Cc1ccc(C2(O)CCC3(CC2)OCCO3)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
HRH3 Q9Y5N1 3/20 0.39
OPRM1 P35372 4/20 0.38
OPRK1 P41145 4/20 0.38
OPRL1 P41146 4/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
C5AR1 P21730 1/20 0.36
ALDH1A1 P00352 2/20 0.35
TSHR P16473 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
HTR1D P28221 1/20 0.34
OPRD1 P41143 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP26A1 O43174 1/20 0.32
CYP26B1 Q9NR63 1/20 0.32
LTA4H P09960 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14403245 0.82 DRD2 (0.39) SLC6A4SLC6A3HRH3OPRM1OPRK1
SCHEMBL8453460 0.80 OPRL1 (0.49) SLC6A4SLC6A3OPRM1OPRK1OPRL1
SCHEMBL615022 0.80 OPRL1 (0.47) SLC6A4SLC6A3OPRM1OPRK1OPRL1
SCHEMBL744179 0.79 SLC6A4 (0.34) SLC6A4SLC6A3HRH3NOS3NOS1
SCHEMBL30406901 0.79 SLC6A4 (0.34) SLC6A4SLC6A3HRH3NOS3NOS1
SCHEMBL8585142 0.79 SLC6A4 (0.44) SLC6A4SLC6A3OPRM1OPRK1OPRL1
SCHEMBL613489 0.77 OPRM1 (0.50) SLC6A4SLC6A3OPRM1OPRK1OPRL1
SCHEMBL8780434 0.75 HRH3 (0.41) HRH3OPRM1OPRK1OPRL1NOS3
SCHEMBL13324152 0.75 OPRL1 (0.47) SLC6A4SLC6A3HRH3OPRM1OPRK1
SCHEMBL613410 0.74 DRD2 (0.55) SLC6A4SLC6A3OPRM1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757669-B1 O-ACYL-4-PHENYL-CYCLOHEXANOLS, THEIR SALTS, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND THEIR USE, AS WELL AS A METHOD OF PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1998-11-18 EP disclosed