SCHEMBL878113

SCHEMBL878113

O=C(O)c1cc2c(cc1F)C(Nc1ccccc1Cl)CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.40
TAS1R1 Q7RTX1 2/20 0.40
TAS1R2 Q8TE23 1/20 0.40
GRIK1 P39086 2/20 0.39
PTK2B Q14289 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DHODH Q02127 1/20 0.37
FABP3 P05413 1/20 0.37
FABP4 P15090 1/20 0.37
FADS1 O60427 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 3/20 0.36
STAT3 P40763 1/20 0.36
STAT1 P42224 1/20 0.36
PBRM1 Q86U86 1/20 0.36
SCN1A P35498 2/20 0.36
SCN5A Q14524 2/20 0.36
SCN8A Q9UQD0 2/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL785625 0.82 ALDH1A1 (0.57) TAS1R3TAS1R1TAS1R2CYP2C19ALDH1A1
SCHEMBL785162 0.82 ALDH1A1 (0.57) TAS1R3TAS1R1TAS1R2CYP2C19ALDH1A1
SCHEMBL878046 0.81 SMN1; SMN2 (0.45) TAS1R3TAS1R1TAS1R2PTK2BSMN1; SMN2
SCHEMBL484460 0.78 ALDH1A1 (0.57) TAS1R3TAS1R1TAS1R2CYP2C19ALDH1A1
SCHEMBL785361 0.78 ALDH1A1 (0.57) TAS1R3TAS1R1TAS1R2CYP2C19ALDH1A1
SCHEMBL883817 0.73 TAS1R3 (0.49) TAS1R3TAS1R1TAS1R2SMN1; SMN2ALDH1A1
SCHEMBL785977 0.72 ACHE (0.37) SMN1; SMN2
SCHEMBL2822056 0.71 ALDH1A1 (0.67) TAS1R3TAS1R1TAS1R2ALDH1A1HTT
SCHEMBL2822060 0.71 ALDH1A1 (0.67) TAS1R3TAS1R1TAS1R2ALDH1A1HTT
SCHEMBL785280 0.70 ALDH1A1 (0.54) TAS1R3TAS1R1TAS1R2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed