SCHEMBL8780919

SCHEMBL8780919

CCN(CCCOc1ccc(N)cc1)CCCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.41
APP P05067 2/20 0.41
KDM4E B2RXH2 1/20 0.40
SIGMAR1 Q99720 1/20 0.38
MAOB P27338 2/20 0.38
PKM P14618 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
MAOA P21397 1/20 0.38
KCNH2 Q12809 1/20 0.38
MCHR1 Q99705 1/20 0.38
XDH P47989 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780789 0.97 ADORA2A (0.41) HRH3APPKDM4EPKMADORA3
SCHEMBL8780940 0.90 ADORA2A (0.43) SIGMAR1PKMADORA3ADORA2AADORA2B
SCHEMBL8780776 0.89 MAOA (0.37) MAOBPKMADORA3ADORA2AADORA2B
SCHEMBL8780869 0.87 KCNH2 (0.42) KDM4EADORA1KCNH2
SCHEMBL8780903 0.86 KCNH2 (0.38) SIGMAR1ADORA1KCNH2
SCHEMBL8780892 0.85 RXFP1 (0.42) HRH3APPADORA3ADORA2AADORA2B
SCHEMBL8780829 0.85 RIPK2 (0.43) HRH3KDM4ESIGMAR1MAOBADORA3
SCHEMBL8780990 0.85 KCNH2 (0.39) PKMADORA3ADORA2AADORA2BADORA1
SCHEMBL8780851 0.85 KCNH2 (0.55) HRH3PKMKCNH2
SCHEMBL8780988 0.84 KCNH2 (0.41) KDM4EADORA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed