SCHEMBL8780776

SCHEMBL8780776

CCCN(CCCc1cc(=O)n(C)c(=O)n1C)CCOc1ccc(N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
PKM P14618 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
KCNH2 Q12809 2/20 0.36
MCHR1 Q99705 1/20 0.36
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CHRM2 P08172 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTR1A P08908 1/20 0.36
GAA P10253 1/20 0.36
CYP2D6 P10635 1/20 0.36
DRD3 P35462 1/20 0.36
SCN1A P35498 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780815 0.93 ADORA2A (0.38) MAOAMAOBPKMADORA3ADORA2A
SCHEMBL8780789 0.92 ADORA2A (0.41) PKMADORA3ADORA2AADORA2BADORA1
SCHEMBL8780919 0.89 HRH3 (0.41) MAOAMAOBPKMADORA3ADORA2A
SCHEMBL8780859 0.86 SLC22A2 (0.42) KCNH2BCHECYP1A2MAPT
SCHEMBL8780802 0.86 L3MBTL1 (0.44) MAOBPKMBCHEACHEGAA
Hydrochloric Acid SCHEMBL8781133 0.85 L3MBTL1 (0.43) MAOBPKMBCHEACHEGAA
SCHEMBL8780890 0.85 PKM (0.52) PKMKCNH2LMNAKMT2A
SCHEMBL8780990 0.85 KCNH2 (0.39) PKMADORA3ADORA2AADORA2BADORA1
SCHEMBL8780940 0.85 ADORA2A (0.43) PKMADORA3ADORA2AADORA2BADORA1
SCHEMBL8780889 0.85 SLC22A2 (0.40) KCNH2CYP3A4CYP2D6DRD3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed