SCHEMBL8780990

SCHEMBL8780990

CN(CCCc1cc(=O)n(C)c(=O)n1C)CCOc1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.39
MCHR1 Q99705 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
PKM P14618 2/20 0.36
CACNA1F O60840 1/20 0.36
CHRM2 P08172 1/20 0.36
ACHE P22303 1/20 0.36
AGTR1 P30556 1/20 0.36
DRD3 P35462 1/20 0.36
CACNA1D Q01668 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
MAPK14 Q16539 1/20 0.36
LTA4H P09960 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780867 0.93 KCNH2 (0.43) KCNH2MCHR1ADORA3ADORA2AADORA2B
SCHEMBL8780781 0.88 LTA4H (0.46) KCNH2MCHR1LTA4HSMN1; SMN2
SCHEMBL8780789 0.86 ADORA2A (0.41) KCNH2MCHR1ADORA3ADORA2AADORA2B
SCHEMBL8780750 0.85 TDP1 (0.37) KCNH2MCHR1ADORA3ADORA2AADORA2B
SCHEMBL8780776 0.85 MAOA (0.37) KCNH2MCHR1ADORA3ADORA2AADORA2B
SCHEMBL8781045 0.85 MAOB (0.49) PKMLTA4HDRD2
SCHEMBL8780919 0.85 HRH3 (0.41) KCNH2MCHR1ADORA3ADORA2AADORA2B
SCHEMBL8780927 0.84 KCNH2 (0.58) KCNH2PKMDRD3SMN1; SMN2DRD2
SCHEMBL8780912 0.84 SIGMAR1 (0.47) KCNH2
SCHEMBL8780850 0.83 KCNH2 (0.59) KCNH2CACNA1FCHRM2ACHEAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed