SCHEMBL878327

SCHEMBL878327

Cc1cc(N2CCC(N(C)C(=O)c3ccc4c(c3)C(N3C=C(OC(=O)O)C(C(F)(F)F)=CC3)CC4)CC2)cc(C)n1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
F10 P00742 1/20 0.33
PDK2 Q15119 1/20 0.32
JAK2 O60674 6/20 0.31
JAK1 P23458 6/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL876437 0.91 F10 (0.33) F10PDK2JAK2JAK1
SCHEMBL876499 0.86 SLC2A1 (0.35) F10PDK2JAK2JAK1
SCHEMBL875680 0.85 F10 (0.33) F10PDK2JAK2JAK1
SCHEMBL877626 0.82 TLR9 (0.37) TLR9TLR8TLR7F10PDK2
SCHEMBL878362 0.79 TLR9 (0.36) TLR9TLR8TLR7F10JAK2
SCHEMBL876160 0.79 F10 (0.33) F10
SCHEMBL878326 0.77 TLR9 (0.39) TLR9TLR8TLR7F10PDK2
SCHEMBL876778 0.75 BDKRB1 (0.39) F10
SCHEMBL876715 0.74 CCR5 (0.37) F10PDK2JAK2JAK1ADORA2A
SCHEMBL785591 0.74 F10 (0.44) TLR9TLR8TLR7F10PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed