SCHEMBL8784649

SCHEMBL8784649

c1ccc(-c2ccc3c(c2)c2ccccc2n3-c2cccc3c2-c2ccccc2C32c3ccccc3-c3c(-n4c5ccccc5c5cc(-c6ccccc6)ccc54)cccc32)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSPO P30536 3/20 0.36
ALDH1A1 P00352 1/20 0.35
PDK2 Q15119 1/20 0.32
DNM1 Q05193 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PDE6D O43924 1/20 0.31
DUSP3 P51452 1/20 0.31
EDNRB P24530 1/20 0.30
EDNRA P25101 1/20 0.30
NPY5R Q15761 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18160225 0.99 TSPO (0.36) TSPOALDH1A1PDK2DNM1KDM4E
SCHEMBL16810702 0.99 TSPO (0.36) TSPOALDH1A1PDK2DNM1KDM4E
SCHEMBL18457743 0.99 TSPO (0.36) TSPOALDH1A1PDK2DNM1KDM4E
SCHEMBL16810747 0.98 TSPO (0.35) TSPOALDH1A1PDK2DNM1KDM4E
SCHEMBL25843929 0.96 TSPO (0.34) TSPOALDH1A1PDK2DNM1
SCHEMBL20232306 0.95 PDK2 (0.35) TSPOPDK2PDE6D
SCHEMBL21138936 0.95 ALDH1A1 (0.33) TSPOALDH1A1KDM4EATML3MBTL1
SCHEMBL21138925 0.95 PDK2 (0.36) TSPOPDK2PDE6D
SCHEMBL15213618 0.95 PDK2 (0.36) TSPOPDK2PDE6D
SCHEMBL18457468 0.94 L3MBTL1 (0.40) TSPOALDH1A1PDK2KDM4EATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8859111-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2014-10-14 US disclosed
US-8859111-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2014-10-14 US disclosed
US-20120126179-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2012-05-24 US disclosed
US-20120126179-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2012-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120126179-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES EPB41, HCN4, EPB41L2 TSPO 991/4885ALDH1A1 327/4885PDK2 1109/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.