SCHEMBL8787115

SCHEMBL8787115

COc1c(Cl)ccnc1OC(=O)NC(=O)CN

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.34
JAK2 O60674 1/20 0.34
TYK2 P29597 1/20 0.34
CARM1 Q86X55 1/20 0.33
KMT2A Q03164 2/20 0.33
P2RX7 Q99572 1/20 0.32
RAF1 P04049 1/20 0.32
MEP1B Q16820 1/20 0.32
POLB P06746 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
BLM P54132 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8785737 0.86 SMN1; SMN2 (0.37) ALDH1A1KDM4EGAATSHRCARM1
SCHEMBL8785157 0.80 FAAH (0.38) KDM4EGAAKMT2ASMN1; SMN2
SCHEMBL8786684 0.79 CYP1A2 (0.39) ALDH1A1KDM4ECARM1SMN1; SMN2
SCHEMBL8786169 0.78 LMNA (0.40) KMT2ASMN1; SMN2
SCHEMBL8785926 0.78 KMT2A (0.40) ALDH1A1GAATSHRKMT2ASMN1; SMN2
SCHEMBL8786282 0.77 CARM1 (0.33) CARM1
SCHEMBL8789020 0.76 CARM1 (0.44) ALDH1A1GAAHSD17B10CARM1KMT2A
SCHEMBL8785043 0.76 NPBWR1 (0.41) ALDH1A1KDM4EGAACARM1KMT2A
SCHEMBL8373693 0.76 ALDH1A1 (0.46) TAS1R3TAS1R1ALDH1A1KDM4ETSHR
Hydrochloric Acid SCHEMBL8786807 0.75 CARM1 (0.43) ALDH1A1GAAHSD17B10CARM1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0650961-B1 Substituted heterocyclic carboxylic acid amides, their preparation, and their use as medicaments HOECHST AG (DE) 1997-03-05 EP disclosed
EP-0650961-A1 Substituted heterocyclic carboxylic acid amides, their preparation, and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-03 EP disclosed