SCHEMBL8788754

SCHEMBL8788754

COc1cccc2c1C(=O)N(CCN1CCC(c3onc4cc(F)ccc34)CC1)C2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.41
HTR2A P28223 4/20 0.41
HTR1A P08908 4/20 0.41
HTR2C P28335 2/20 0.41
ABCB11 O95342 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRA2A P08913 1/20 0.40
CHRM1 P11229 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
ACHE P22303 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
CCKBR P32239 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787429 0.87 DRD2 (0.47) DRD2HTR2AHTR1AHTR2CACHE
Hydrochloric Acid SCHEMBL8787530 0.86 DRD2 (0.46) DRD2HTR2AHTR1AHTR2CACHE
SCHEMBL8787720 0.85 ACHE (0.47) DRD2HTR2AHTR1AACHE
SCHEMBL1545035 0.85 ACHE (0.60) DRD2HTR2AHTR1AHTR2CABCB11
SCHEMBL7773189 0.84 DRD2 (0.46) DRD2HTR2AHTR1AHTR2CACHE
Hydrochloric Acid SCHEMBL1545060 0.84 ACHE (0.59) DRD2HTR2AHTR1AHTR2CABCB11
SCHEMBL8789443 0.84 ACHE (0.46) DRD2HTR2AHTR1AACHESLC6A4
SCHEMBL8863522 0.84 ACHE (0.46) DRD2HTR2AHTR1AHTR2CACHE
SCHEMBL8788723 0.82 DRD2 (0.49) DRD2HTR2AHTR1AHTR2CDRD4
SCHEMBL9096725 0.82 ACHE (0.44) DRD2HTR2AHTR1AACHESLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed