SCHEMBL8788375

SCHEMBL8788375

CC(C)(O)CCN1CCC(c2snc3cc(F)ccc23)CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.40
SLC6A4 P31645 4/20 0.40
HTR2A P28223 7/20 0.40
HTR7 P34969 5/20 0.40
KCNH2 Q12809 4/20 0.40
ACHE P22303 2/20 0.39
DRD3 P35462 2/20 0.36
HTR4 Q13639 1/20 0.36
ADRA1D P25100 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8788085 0.89 DRD2 (0.41) DRD2SLC6A4HTR2AHTR7KCNH2
SCHEMBL1545159 0.80 HTR1D (0.52) DRD2SLC6A4HTR2AHTR7KCNH2
SCHEMBL8788384 0.79 CCR3 (0.44) DRD2SLC6A4HTR2AHTR7KCNH2
SCHEMBL8788032 0.78 DRD2 (0.47) DRD2SLC6A4HTR2AHTR7KCNH2
SCHEMBL8787809 0.76 HTR1A (0.41) DRD2HTR2AHTR7ACHE
SCHEMBL8789213 0.76 DRD2 (0.43) DRD2SLC6A4HTR2AHTR7ACHE
SCHEMBL1545719 0.74 DRD2 (0.74) DRD2SLC6A4HTR2AHTR7KCNH2
Hydrochloric Acid SCHEMBL9231660 0.73 DRD2 (0.45) DRD2SLC6A4HTR2AHTR7KCNH2
SCHEMBL7769075 0.72 HTR1A (0.49) DRD2SLC6A4HTR2AKCNH2ACHE
SCHEMBL1545221 0.70 HTR1D (0.51) DRD2SLC6A4HTR2AHTR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP claimed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP claimed