SCHEMBL8788384

SCHEMBL8788384

CCOC(=O)CCN1CCC(c2snc3cc(F)ccc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 3/20 0.44
ALDH1A1 P00352 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
DRD2 P14416 8/20 0.41
HTR2A P28223 8/20 0.41
HTR7 P34969 8/20 0.41
KCNH2 Q12809 7/20 0.41
KDM4E B2RXH2 2/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
SLC6A4 P31645 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545311 0.82 HTR1D (0.53) CCR3ALDH1A1TDP1DRD2HTR2A
Hydrochloric Acid SCHEMBL7722897 0.82 HTR1D (0.52) CCR3ALDH1A1TDP1DRD2HTR2A
SCHEMBL8788170 0.80 HTR2A (0.47) CCR3DRD2HTR2AHTR7KCNH2
SCHEMBL8788085 0.79 DRD2 (0.41) DRD2HTR2AHTR7KCNH2SLC6A4
SCHEMBL8788375 0.79 DRD2 (0.40) DRD2HTR2AHTR7KCNH2SLC6A4
SCHEMBL21034705 0.77 IDO1 (0.49) DRD2KCNH2CYP3A4SLC6A4
SCHEMBL1545575 0.77 DRD2 (0.70) DRD2HTR2AHTR7KCNH2SLC6A4
SCHEMBL6994781 0.76 DRD2 (0.53) ALDH1A1TDP1DRD2HTR2AKDM4E
SCHEMBL8787809 0.74 HTR1A (0.41) DRD2HTR2AHTR7
SCHEMBL8789213 0.74 DRD2 (0.43) DRD2HTR2AHTR7SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP claimed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP claimed
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed