SCHEMBL8788929

SCHEMBL8788929

CC(=O)NCCNc1ccc(NCCNC(C)=O)c2c1C(=O)c1ccncc1C2=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.58
MUS81 Q96NY9 1/20 0.58
BLM P54132 4/20 0.45
MEN1 O00255 1/20 0.45
NSD2 O96028 1/20 0.45
POLB P06746 1/20 0.45
KMT2A Q03164 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
TOP2B Q02880 1/20 0.44
CYP3A4 P08684 10/20 0.42
TP53 P04637 3/20 0.42
MAPT P10636 3/20 0.42
CASP1 P29466 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
CASP7 P55210 2/20 0.42
HSD17B10 Q99714 5/20 0.42
CYP1A2 P05177 5/20 0.42
ALOX15 P16050 4/20 0.42
TSHR P16473 4/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8788938 0.83 ECE1 (0.57) ECE1MUS81BLMMEN1NSD2
SCHEMBL7766945 0.83 ECE1 (0.53) ECE1MUS81BLMMEN1NSD2
SCHEMBL8788985 0.83 ECE1 (0.55) ECE1MUS81BLMMEN1NSD2
Hydrochloric Acid SCHEMBL8788992 0.82 ECE1 (0.56) ECE1MUS81BLMMEN1NSD2
SCHEMBL8788420 0.82 BLM (0.61) ECE1MUS81BLMMEN1NSD2
SCHEMBL8789454 0.81 ECE1 (0.58) ECE1MUS81BLMMEN1NSD2
SCHEMBL8789103 0.81 ECE1 (0.55) ECE1MUS81BLMMEN1NSD2
SCHEMBL8788385 0.80 TOP2B (0.70) ECE1MUS81BLMMEN1NSD2
SCHEMBL8788424 0.80 ECE1 (0.63) ECE1MUS81BLMMEN1NSD2
SCHEMBL8789428 0.80 ECE1 (0.62) ECE1MUS81BLMMEN1NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP claimed
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP disclosed
EP-0575526-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1993-12-29 EP disclosed
WO-1992015300-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO[g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1992-09-17 WO disclosed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP disclosed