SCHEMBL8788985

SCHEMBL8788985

N=C(N)NCCNc1ccc(NCCNC(=N)N)c2c1C(=O)c1ccncc1C2=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.55
MUS81 Q96NY9 1/20 0.55
TOP2B Q02880 1/20 0.43
BLM P54132 9/20 0.41
MAPT P10636 8/20 0.41
SMN1; SMN2 Q16637 7/20 0.41
TP53 P04637 6/20 0.41
CYP3A4 P08684 4/20 0.41
CASP1 P29466 3/20 0.41
CASP7 P55210 2/20 0.41
MEN1 O00255 6/20 0.41
KMT2A Q03164 6/20 0.41
POLB P06746 4/20 0.41
NSD2 O96028 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
CDC25B P30305 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8788929 0.83 ECE1 (0.58) ECE1MUS81TOP2BBLMMAPT
SCHEMBL8789428 0.81 ECE1 (0.62) ECE1MUS81TOP2BBLMMAPT
SCHEMBL8788420 0.81 BLM (0.61) ECE1MUS81TOP2BBLMMAPT
Pixantrone SCHEMBL7825 0.81 ECE1 (0.72) ECE1MUS81TOP2BBLMMAPT
Pixantrone SCHEMBL29372192 0.81 ECE1 (0.72) ECE1MUS81TOP2BBLMMAPT
SCHEMBL8788920 0.80 ECE1 (0.61) ECE1MUS81TOP2BBLMMAPT
Pixantrone SCHEMBL7771183 0.80 ECE1 (0.70) ECE1MUS81TOP2BBLMMAPT
SCHEMBL8788938 0.80 ECE1 (0.57) ECE1MUS81TOP2BBLMMAPT
Pixantrone SCHEMBL17673194 0.80 ECE1 (0.70) ECE1MUS81TOP2BBLMMAPT
SCHEMBL8788385 0.79 TOP2B (0.70) ECE1MUS81TOP2BBLMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP claimed
EP-0575526-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1993-12-29 EP claimed
WO-1992015300-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO[g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1992-09-17 WO claimed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP claimed
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP disclosed
EP-0575526-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1993-12-29 EP disclosed
WO-1992015300-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO[g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1992-09-17 WO disclosed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP disclosed