SCHEMBL8788976

SCHEMBL8788976

CC(N)Nc1ccc(NC(C)N)c2c1C(=O)c1ccncc1C2=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
ECE1 P42892 1/20 0.47
MUS81 Q96NY9 1/20 0.47
CDC25B P30305 1/20 0.46
MAPT P10636 4/20 0.45
TP53 P04637 3/20 0.45
CYP3A4 P08684 3/20 0.45
CASP1 P29466 3/20 0.45
BLM P54132 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
CASP7 P55210 2/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
KDM4E B2RXH2 1/20 0.44
AOC1 P19801 2/20 0.36
AOC3 Q16853 2/20 0.36
CCNE2 O96020 1/20 0.36
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8788434 0.84 MAOA (0.47) MAOAMAOBECE1MUS81CDC25B
SCHEMBL8789326 0.82 MAOA (0.45) MAOAMAOBECE1MUS81CDC25B
SCHEMBL8792588 0.81 ECE1 (0.45) MAOAMAOBECE1MUS81CDC25B
SCHEMBL4198601 0.80 MAPT (0.46) MAOAMAOBCDC25BMAPTCYP3A4
SCHEMBL4193002 0.79 THRB (0.33) MAPTBLMSMN1; SMN2MAPK1CCNE2
Pixantrone SCHEMBL7825 0.74 ECE1 (0.72) MAOAMAOBECE1MUS81CDC25B
Pixantrone SCHEMBL29372192 0.74 ECE1 (0.72) MAOAMAOBECE1MUS81CDC25B
SCHEMBL8789103 0.74 ECE1 (0.55) MAOAMAOBECE1MUS81CDC25B
SCHEMBL8788509 0.74 ECE1 (0.52) MAOAMAOBECE1MUS81CDC25B
Pixantrone SCHEMBL17673194 0.73 ECE1 (0.70) MAOAMAOBECE1MUS81CDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP disclosed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP disclosed