SCHEMBL8790260

SCHEMBL8790260

CCCS(=O)(=O)CCCCCCCCCCCCc1c(O)ccc2[nH]c(-c3ccc(O)cc3)c(C)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.39
ESR2 Q92731 4/20 0.39
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CCNB2 O95067 3/20 0.38
CDK1 P06493 3/20 0.38
CCNB1 P14635 3/20 0.38
GSK3A P49840 3/20 0.38
GSK3B P49841 3/20 0.38
CDK5 Q00535 3/20 0.38
CDK5R1 Q15078 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7692326 0.97 ESR1 (0.43) ESR1ESR2MAPK1KDM4EALDH1A1
SCHEMBL8789363 0.85 MAPK1 (0.36) ESR1ESR2MAPK1KDM4EALDH1A1
SCHEMBL8790299 0.81 CCNB2 (0.41) ESR1ESR2MAPK1KDM4EALDH1A1
SCHEMBL9356958 0.80 NR1I2 (0.40) MAPK1CCNB2CDK1CCNB1GSK3A
SCHEMBL8792445 0.80 CCNB2 (0.38) ESR1MAPK1KDM4EALDH1A1HPGD
SCHEMBL8789330 0.80 CCNB2 (0.40) ESR1MAPK1KDM4EALDH1A1HPGD
SCHEMBL8789465 0.79 CCNB2 (0.42) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL9027686 0.79 ALDH1A1 (0.39) MAPK1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9027574 0.76 DRD2 (0.39) MAPK1CCNB2CDK1CCNB1GSK3A
SCHEMBL9028366 0.75 CCNB2 (0.38) MAPK1CCNB2CDK1CCNB1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772591-A1 2-PHENYL INDOLES AS ANTI-OESTROGEN DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-14 EP disclosed
WO-1996003375-A1 2-PHENYL INDOLES AS ANTI-OESTROGEN DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1996-02-08 WO disclosed