SCHEMBL8792218

SCHEMBL8792218

COc1cccc(C23CCN(Cc4ccccc4)CC2CCC(=O)C3)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.56
OPRD1 P41143 2/20 0.56
OPRK1 P41145 2/20 0.56
SIGMAR1 Q99720 5/20 0.48
CXCR3 P49682 2/20 0.48
CHRM2 P08172 1/20 0.47
CHRM3 P20309 1/20 0.47
ALDH1A1 P00352 1/20 0.46
SLC6A4 P31645 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8793354 0.90 OPRM1 (0.55) OPRM1OPRD1OPRK1SIGMAR1SLC6A4
SCHEMBL8395140 0.88 OPRM1 (0.57) OPRM1OPRD1OPRK1CXCR3CHRM2
SCHEMBL8395142 0.88 OPRM1 (0.57) OPRM1OPRD1OPRK1CXCR3CHRM2
SCHEMBL7486456 0.88 OPRM1 (0.60) OPRM1OPRD1OPRK1SIGMAR1CXCR3
SCHEMBL7486453 0.88 OPRM1 (0.60) OPRM1OPRD1OPRK1SIGMAR1CXCR3
Hydrochloric Acid SCHEMBL7487249 0.87 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1CXCR3
Hydrochloric Acid SCHEMBL7487248 0.87 OPRM1 (0.59) OPRM1OPRD1OPRK1SIGMAR1CXCR3
SCHEMBL8396855 0.86 OPRD1 (0.76) OPRM1OPRD1OPRK1SIGMAR1CXCR3
SCHEMBL11398571 0.86 OPRD1 (0.76) OPRM1OPRD1OPRK1SIGMAR1CXCR3
SCHEMBL8396856 0.86 OPRD1 (0.76) OPRM1OPRD1OPRK1SIGMAR1CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0485636-B1 INDOLE DERIVATIVE TORAY INDUSTRIES (JP) 1997-03-12 EP disclosed
EP-0735026-A1 Method for the production of isoquinoline derivatives and their use as intermediates in the preparation of indole derivatives TORAY INDUSTRIES, INC. (JP) 1996-10-02 EP disclosed
US-5539119-A MULTISTAGE FORMATION BY OXIDATION, REDUCING A CARBAMATE TO FORM AN ENAMINE, FORMING AN OXIDE TORAY INDUSTRIES, INC. (JP) 1996-07-23 US disclosed
US-5244904-A Immunorepressant, analgesic TORAY INDUSTRIES, INC. (JP) 1993-09-14 US disclosed
EP-0485636-A1 INDOLE DERIVATIVE TORAY INDUSTRIES, INC. (JP) 1992-05-20 EP disclosed