SCHEMBL8792437

SCHEMBL8792437

COC(=O)c1sccc1-c1ccc(C)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
MAPT P10636 3/20 0.57
MAPK1 P28482 2/20 0.57
TSHR P16473 2/20 0.57
HSD17B10 Q99714 1/20 0.57
PKM P14618 1/20 0.55
ATM Q13315 1/20 0.55
NPSR1 Q6W5P4 3/20 0.52
POLB P06746 2/20 0.51
KDM4E B2RXH2 1/20 0.51
GABRA1 P14867 1/20 0.51
GABRG2 P18507 1/20 0.51
GABRB3 P28472 1/20 0.51
GABRA5 P31644 1/20 0.51
GABRA3 P34903 1/20 0.51
LMNA P02545 1/20 0.49
PTGS1 P23219 1/20 0.48
HPGD P15428 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20262093 0.87 PTGS1 (0.62) ALDH1A1MAPTNPSR1POLBKDM4E
SCHEMBL6229196 0.85 GABRA1 (0.67) ALDH1A1MAPTNPSR1POLBKDM4E
SCHEMBL13098291 0.81 MAPK10 (0.56) ALDH1A1MAPTMAPK1HSD17B10NPSR1
SCHEMBL8791515 0.81 KDM4E (0.53) ALDH1A1MAPTMAPK1TSHRHSD17B10
SCHEMBL28208998 0.81 HSD17B10 (0.61) ALDH1A1MAPTHSD17B10PKMATM
SCHEMBL1339762 0.81 BCAT2 (0.51) ALDH1A1MAPTMAPK1TSHRHSD17B10
SCHEMBL2231308 0.79 BCAT2 (0.69) ALDH1A1MAPTMAPK1TSHRHSD17B10
SCHEMBL24611525 0.79 KDM4E (0.50) ALDH1A1MAPTTSHRHSD17B10NPSR1
Potassium Ion SCHEMBL28679802 0.78 PTGS2 (0.46) ALDH1A1MAPTMAPK1TSHRHSD17B10
SCHEMBL15940088 0.78 MAPT (0.67) ALDH1A1MAPTMAPK1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849035-A Phenyl heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2018-03-27 CN disclosed
EP-0783518-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO. INC. (US) 1997-07-16 EP disclosed
EP-0652869-B1 IMIDAZOLE ETHERS HAVING A II ANTAGONIST ACTIVITY LUSO FARMACO INST (IT) 1997-03-26 EP disclosed
EP-0652869-A1 IMIDAZOLE ETHERS HAVING A II ANTAGONIST ACTIVITY. LUSO FARMACO INST (IT) 1995-05-17 EP disclosed
WO-1994002467-A1 IMIDAZOLE ETHERS HAVING A II ANTAGONIST ACTIVITY INSTITUTO LUSO FARMACO D'ITALIA S.P.A. (IT) 1994-02-03 WO disclosed