SCHEMBL8795010

SCHEMBL8795010

CC1(C)C=C(C(N)=NC#N)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.36
MAPT P10636 7/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MCL1 Q07820 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
ABCC9 O60706 1/20 0.33
ALDH1A1 P00352 4/20 0.33
AKR1B1 P15121 2/20 0.33
MAPK1 P28482 1/20 0.33
HPRT1 P00492 1/20 0.33
NOS1 P29475 2/20 0.33
CYP3A4 P08684 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8793999 0.84 EGFR (0.34) EGFRMAPTKDM4ECA1CA2
SCHEMBL8795895 0.84 EGFR (0.34) EGFRMAPTKDM4EMEN1KMT2A
SCHEMBL29442980 0.84 EGFR (0.34) EGFRMAPTKDM4ECA1CA2
SCHEMBL8794980 0.82 ALDH1A1 (0.36) EGFRMAPTKDM4EMEN1KMT2A
SCHEMBL8794987 0.82 ALDH1A1 (0.36) EGFRMAPTKDM4EMEN1KMT2A
SCHEMBL27328716 0.81 CA1 (0.38) MAPTKDM4EMEN1KMT2AMCL1
SCHEMBL27316930 0.81 PRSS1 (0.40) MAPTKDM4EMEN1KMT2AMCL1
SCHEMBL8795381 0.80 KMT2A (0.38) EGFRMAPTKDM4EMEN1KMT2A
SCHEMBL8308734 0.78 AKR1B1 (0.43) MAPTMEN1KMT2ACA1CA2
SCHEMBL8794821 0.78 VCAM1 (0.40) EGFRCA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0541807-B1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1997-12-17 EP disclosed
US-5412117-A Potassium channel activators, antiasmatics, antiepileptics CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-05-02 US disclosed
EP-0541807-A1 NOVEL BENZOPYRAN DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 1993-05-19 EP disclosed