SCHEMBL8795276

SCHEMBL8795276

CC1=CN(c2ccc(-c3ccc(C(=O)Nc4ccc5ccn(CCN(C)C)c5c4)cc3)c(C)c2)NO1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.44
HTR1B P28222 5/20 0.44
HTR2A P28223 5/20 0.44
EPHX2 P34913 2/20 0.40
NR1H4 Q96RI1 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CHRM2 P08172 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7935768 0.79 HTR1D (0.65) HTR1DHTR1BHTR2AEPHX2NR1H4
SCHEMBL8792134 0.78 HTR1D (0.59) HTR1DHTR1BHTR2AKDM4EMEN1
SCHEMBL1122381 0.66 ALDH1A1 (0.53) HTR1DHTR2AALDH1A1MAPTHPGD
SCHEMBL8615090 0.65 HTR6 (0.49) HTR1DHTR1BHTR2AKDM4EMAPT
SCHEMBL8795470 0.64 HTR1D (0.62) HTR1DHTR1BHTR2AKDM4EMEN1
SCHEMBL1122080 0.64 HTR2A (0.53) HTR1DHTR2AHTR2CHTR6
SCHEMBL30443765 0.63 HTR2C (0.58) HTR1DHTR2AHTR2CHTR6
SCHEMBL5244630 0.62 MAPT (0.53) HTR1DHTR1BHTR2AKDM4EMEN1
SCHEMBL1122382 0.62 HTR6 (0.51) HTR1DHTR2AEPHX2NR1H4HTR2C
Hydrochloric Acid SCHEMBL5249374 0.62 MAPT (0.52) HTR1DHTR1BHTR2AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0763034-A1 AMIDE DERIVATIVES HAVING 5HT1D-ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1997-03-19 EP disclosed
WO-1995032967-A1 AMIDE DERIVATIVES HAVING 5HT1D-ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-12-07 WO disclosed