SCHEMBL8795459

SCHEMBL8795459

CCOC(=O)CCCCC(=O)c1ccc(OC)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 3/20 0.62
WNT3A P56704 3/20 0.62
TSHR P16473 2/20 0.55
MAPT P10636 1/20 0.55
PAX8 Q06710 1/20 0.52
MAPK1 P28482 1/20 0.51
ALDH1A1 P00352 3/20 0.51
CYP2C19 P33261 2/20 0.51
POLB P06746 1/20 0.51
PDE4B Q07343 3/20 0.50
PDE4A P27815 2/20 0.50
PDE4C Q08493 2/20 0.50
PDE4D Q08499 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TNF P01375 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11705162 0.91 CTNNB1 (0.70) CTNNB1WNT3ATSHRMAPTPAX8
SCHEMBL31556192 0.88 CTNNB1 (0.73) CTNNB1WNT3ATSHRMAPTPAX8
SCHEMBL31556194 0.86 CTNNB1 (0.71) CTNNB1WNT3ATSHRMAPTPAX8
SCHEMBL3814415 0.85 THRA (0.59) CTNNB1WNT3ATSHRMAPK1PDE4B
SCHEMBL9375696 0.85 CTNNB1 (0.65) CTNNB1WNT3ATSHRMAPTALDH1A1
SCHEMBL9119840 0.85 CTNNB1 (0.65) CTNNB1WNT3ATSHRMAPTPAX8
SCHEMBL20009310 0.84 KMT2A (0.60) CTNNB1WNT3ATSHRMAPTMAPK1
SCHEMBL2848397 0.84 MEN1 (0.70) CTNNB1WNT3ATSHRMAPTMAPK1
SCHEMBL31314527 0.84 MEN1 (0.70) CTNNB1WNT3ATSHRMAPTMAPK1
SCHEMBL5355533 0.84 CTNNB1 (0.63) CTNNB1WNT3ATSHRMAPTPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634401-B1 MDR reversal agents AMERICAN CYANAMID CO (US) 1997-08-13 EP disclosed
US-5639887-A MULTIDRUG RESISTANT CELLS; INCREASE CELL SENSITIVITY TO ANTICANCER AGENTS AMERICAN CYANAMID COMPANY (US) 1997-06-17 US disclosed
US-5561141-A POTENTIATE ACTIVITY OF ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY (US) 1996-10-01 US disclosed
US-5550149-A SULFUR-CONTAINING COMPOUNDS THAT ARE EFFECTIVE IN POTENTIATING THE ACTIVITY OF CHEMOTHERAPEUTIC ANTI-CANCER AGENTS BY INCREASING SENSITIVITY OF MULTI-DRUG RESISTANT CELLS AMERICAN CYANAMID COMPANY (US) 1996-08-27 US disclosed
US-5387685-A MDR reversal agents AMERICAN CYANAMID COMPANY 1995-02-07 US disclosed
EP-0634401-A1 MDR reversal agents AMERICAN CYANAMID COMPANY (US) 1995-01-18 EP disclosed