SCHEMBL8796969

SCHEMBL8796969

O=C1NC(Cc2ccc(OCCN3COc4ccc(C(F)(F)F)cc4C3=O)cc2)C(=O)S1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 3/20 0.36
KCNH2 Q12809 2/20 0.35
MCHR1 Q99705 1/20 0.35
PSEN1 P49768 3/20 0.34
PSEN2 P49810 3/20 0.34
APH1B Q8WW43 3/20 0.34
NCSTN Q92542 3/20 0.34
APH1A Q96BI3 3/20 0.34
PSENEN Q9NZ42 3/20 0.34
HRH3 Q9Y5N1 5/20 0.33
PTPN1 P18031 1/20 0.33
GHSR Q92847 1/20 0.32
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
LTA4H P09960 1/20 0.31
TNIK Q9UKE5 1/20 0.31
SCN1A P35498 1/20 0.31
SCN4A P35499 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797588 0.89 DRD2 (0.36) KCNH2MCHR1HRH3MAOAMAOB
SCHEMBL8797133 0.87 HRH3 (0.34) FFAR1HRH3
SCHEMBL8797688 0.87 HRH3 (0.35) FFAR1HRH3
SCHEMBL8796797 0.87 FFAR1 (0.39) FFAR1KCNH2MCHR1PSEN1PSEN2
SCHEMBL8797138 0.87 HRH3 (0.34) FFAR1HRH3
SCHEMBL8796803 0.86 HTT (0.36) HRH3
SCHEMBL8797429 0.86 MAOB (0.35) FFAR1HRH3MAOAMAOBTNIK
SCHEMBL8797111 0.85 HRH3 (0.35) FFAR1HRH3TNIK
SCHEMBL8797027 0.85 HRH3 (0.36) FFAR1HRH3MAOB
SCHEMBL8797744 0.85 HRH3 (0.35) FFAR1HRH3MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787727-A1 Benzoazine derivative or salt thereof and pharmaceutical composition comprising the same SS Pharmaceutical Co., Ltd. (JP) 1997-08-06 EP disclosed