SCHEMBL8798376

SCHEMBL8798376

COC(=O)c1c(-c2cccc(C)c2)ccnc1NC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.50
ALDH1A1 P00352 4/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
MAPK14 Q16539 1/20 0.41
TOP2A P11388 2/20 0.40
KMO O15229 1/20 0.40
ADORA2A P29274 1/20 0.39
BDKRB1 P46663 2/20 0.39
KDM4E B2RXH2 3/20 0.39
LMNA P02545 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SYK P43405 1/20 0.39
JMJD6 Q6NYC1 1/20 0.39
POLQ O75417 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443036 0.88 KMO (0.47) HSD17B10ALDH1A1KMT2AMAPTMEN1
SCHEMBL21749975 0.72 MAPT (0.39) ALDH1A1KMT2AMAPTMEN1KDM4E
SCHEMBL23201168 0.72 ALDH1A1 (0.51) HSD17B10ALDH1A1KMT2AMAPTMAPK14
SCHEMBL25586500 0.69 HSD17B10 (0.47) HSD17B10MAPK14ADORA2A
SCHEMBL11821346 0.69 KMO (0.51) HSD17B10ALDH1A1KMT2AMAPTKMO
SCHEMBL28493467 0.69 KDM4E (0.60) MAPK14KMOKDM4ESYKJMJD6
SCHEMBL3515932 0.68 BDKRB1 (0.42) HSD17B10ALDH1A1MAPTTOP2ABDKRB1
SCHEMBL30285097 0.67 SLC6A3 (0.63) HSD17B10ALDH1A1KMT2AMAPTMEN1
SCHEMBL3516370 0.67 GABRG2 (0.39) HSD17B10ALDH1A1MAPTBDKRB1KDM4E
SCHEMBL13521521 0.67 CCNT1 (0.61) HSD17B10ALDH1A1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804438-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-11-05 EP disclosed