SCHEMBL8798451

SCHEMBL8798451

O=C(O)CC(CC(=O)O)c1ccc2c(c1)OCO2.O=C1CC(c2ccc3c(c2)OCO3)CC(=O)O1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
MAPT P10636 5/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
HPGD P15428 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
NPC1 O15118 1/20 0.45
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
MAPK9 P45984 1/20 0.43
KDM4E B2RXH2 1/20 0.39
MCL1 Q07820 1/20 0.39
TSHR P16473 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
CYP2C9 P11712 1/20 0.39
HSD17B2 P37059 1/20 0.39
ALOX15B O15296 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5858099 0.83 KMT2A (0.62) ALDH1A1KMT2AL3MBTL1CYP1A2CYP2C19
SCHEMBL5856811 0.81 ALDH1A1 (0.60) ALDH1A1MAPTKMT2AMEN1HPGD
SCHEMBL8798404 0.79 PRKCZ (0.40) ALDH1A1KMT2AMEN1CYP1A2CYP2C19
SCHEMBL5847436 0.76 KMT2A (0.55) ALDH1A1KMT2AMEN1L3MBTL1CYP1A2
SCHEMBL8798443 0.75 KMT2A (0.57) ALDH1A1KMT2AMEN1L3MBTL1CYP1A2
SCHEMBL6219736 0.75 KMT2A (0.54) ALDH1A1KMT2AMEN1HPGDL3MBTL1
SCHEMBL7815155 0.75 KMT2A (0.57) ALDH1A1KMT2AMEN1L3MBTL1CYP1A2
SCHEMBL5847398 0.75 KMT2A (0.54) ALDH1A1KMT2AMEN1L3MBTL1CYP1A2
SCHEMBL20379845 0.74 PTGS1 (0.59) ALDH1A1MAPTKMT2AMEN1HPGD
SCHEMBL20380123 0.73 ALDH1A1 (0.49) ALDH1A1MAPTKMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1085661-C Piperidine derivatives as neurokinin antagonists SCHERING CORP (US) 2002-05-29 CN disclosed
CN-1161033-A Piperidine derivatives as neurokinin antagonists SCHERING CORP (US) 1997-10-01 CN disclosed
EP-0773929-A1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1997-05-21 EP disclosed
WO-1996039386-A1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1996-12-12 WO disclosed