SCHEMBL8798404

SCHEMBL8798404

O=C(O)CC(CC(=O)O)c1ccc(Cl)c(Cl)c1.O=C1CC(c2ccc(Cl)c(Cl)c2)CC(=O)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 2/20 0.40
CYP26A1 O43174 2/20 0.37
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
HSD17B2 P37059 1/20 0.35
GABBR2 O75899 3/20 0.35
GABBR1 Q9UBS5 3/20 0.35
LMNA P02545 2/20 0.35
CYP2C9 P11712 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
NFKB1 P19838 1/20 0.35
DRD3 P35462 1/20 0.35
BLM P54132 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811407 0.86 FNTA (0.38) FNTAFNTBHSD17B2LMNAALDH1A1
SCHEMBL8799604 0.83 FNTA (0.42) FNTAFNTBLMNAALDH1A1CYP3A4
SCHEMBL657183 0.80 SLC6A2 (0.44) CYP2D6THRBSLC6A2SLC6A4SLC6A3
SCHEMBL8798451 0.79 ALDH1A1 (0.46) HSD17B2CYP2C9ALDH1A1CYP1A2CYP2C19
SCHEMBL1532918 0.79 PRKCZ (0.54) PRKCZCYP26A1FNTAFNTBGABBR2
SCHEMBL7815285 0.79 LMNA (0.37) LMNAALDH1A1FFAR1
SCHEMBL657182 0.71 PRKCZ (0.48) PRKCZCYP26A1FNTAFNTBGABBR2
SCHEMBL8798403 0.71 PRKCZ (0.48) PRKCZCYP26A1FNTAFNTBGABBR2
SCHEMBL7633288 0.70 GABBR2 (0.68) PRKCZGABBR2GABBR1LMNACYP2C9
Hydrochloric Acid SCHEMBL560490 0.69 GABBR2 (0.66) PRKCZGABBR2GABBR1LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-A1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1997-05-21 EP disclosed
WO-1996039386-A1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1996-12-12 WO disclosed