SCHEMBL8798488

SCHEMBL8798488

CCOC(=O)OC1Cc2c[nH]c3cccc(c23)C(=O)N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.44
HTR2A P28223 6/20 0.42
HTR2C P28335 4/20 0.42
HTR1A P08908 3/20 0.42
HTR2B P41595 3/20 0.42
HTR6 P50406 3/20 0.42
HTR7 P34969 2/20 0.42
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
KDM4E B2RXH2 5/20 0.41
MAPT P10636 4/20 0.41
RECQL P46063 2/20 0.41
USP2 O75604 2/20 0.41
PLEC Q15149 1/20 0.41
DRD3 P35462 3/20 0.41
ADRB2 P07550 2/20 0.41
ADRB1 P08588 2/20 0.41
DRD2 P14416 2/20 0.41
DRD4 P21917 2/20 0.41
HRH1 P35367 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9483531 0.73 PARP1 (0.54) PARP1HTR2AHTR2CHTR1AHTR2B
SCHEMBL8798234 0.73 PRKCD (0.58) PARP1HTR2AHTR2CHTR1AHTR2B
SCHEMBL8798803 0.70 PARP1 (0.54) PARP1HTR2AHTR2CHTR1AHTR2B
SCHEMBL3043496 0.70 MAPT (0.45) KDM4EMAPTALDH1A1TSHRCYP2C19
Hydrochloric Acid SCHEMBL8798710 0.69 PARP1 (0.52) PARP1HTR2AHTR2CHTR1AHTR2B
Hydrochloric Acid SCHEMBL3052246 0.69 MAPT (0.44) KDM4EMAPTALDH1A1TSHRCYP2C19
SCHEMBL9485325 0.69 PARP1 (0.51) PARP1HTR2AHTR2CHTR1AHTR2B
SCHEMBL8800099 0.68 PARP1 (0.50) PARP1HTR2AHTR2CHTR1AHTR2B
SCHEMBL9483532 0.67 PARP1 (0.42) PARP1HTR2AHTR2CHTR1AHTR2B
SCHEMBL8799119 0.67 PARP1 (0.37) PARP1HTR2AHTR2CHTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525584-B1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them SOLVAY PHARM GMBH (DE) 1997-12-10 EP disclosed
EP-0525584-A1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them Kali-Chemie Pharma GmbH (DE) 1993-02-03 EP disclosed