SCHEMBL8799459

SCHEMBL8799459

CSc1ccc(OC(C)C)c([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.55
XDH P47989 1/20 0.43
CYP19A1 P11511 2/20 0.39
TDP1 Q9NUW8 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
FBP1 P09467 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27028620 0.86 PDK1 (0.41) PDK1MEN1KMT2AMAPTLMNA
SCHEMBL8798263 0.79 PDK1 (0.58) PDK1XDHTDP1MEN1KMT2A
SCHEMBL6809251 0.79 PDK1 (0.58) PDK1CYP19A1TDP1MEN1KMT2A
SCHEMBL29749825 0.79 PDK1 (0.58) PDK1CYP19A1TDP1MEN1KMT2A
SCHEMBL8799454 0.78 ALDH1A1 (0.39) PDK1MEN1KMT2AMAPTLMNA
SCHEMBL16958967 0.78 PDK1 (0.57) PDK1XDHCYP19A1TDP1MEN1
SCHEMBL19175613 0.78 PDK1 (0.61) PDK1XDHKMT2AMAPTNPC1
SCHEMBL14136388 0.78 PDK1 (0.57) PDK1XDHCYP19A1TDP1MEN1
SCHEMBL3043316 0.78 PDK1 (0.57) PDK1XDHCYP19A1TDP1MEN1
SCHEMBL1136078 0.78 PDK1 (0.57) PDK1XDHCYP19A1TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025051129-A1 ARYL HETEROCYCLIC SLC7A11 INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海深势唯思科技有限责任公司 2025-03-13 WO disclosed
CN-119552124-A Aryl heterocycle SLC7A11 inhibitor and preparation method and application thereof 上海深势唯思科技有限责任公司 2025-03-04 CN disclosed
EP-0482771-B1 Heterocyclic acids ZENECA LTD (GB) 1997-06-18 EP disclosed
US-5410064-A Thromboxane A2 antagonists and inhibitors of thromboxane A2 synthase IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-04-25 US disclosed
US-5219874-A Heterocyclic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-06-15 US disclosed
EP-0482771-A2 Heterocyclic acids ZENECA LIMITED (GB) 1992-04-29 EP disclosed