SCHEMBL8799536

SCHEMBL8799536

NCC(=O)NS(=O)(=O)c1nc2ccccc2s1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.70
CA2 P00918 7/20 0.70
CA12 O43570 1/20 0.55
CA4 P22748 1/20 0.55
CA7 P43166 1/20 0.55
CA14 Q9ULX7 1/20 0.55
PSMB8 P28062 1/20 0.53
PSMB5 P28074 1/20 0.53
ALDH1A1 P00352 5/20 0.48
MAPT P10636 3/20 0.48
LMNA P02545 2/20 0.48
HTT P42858 2/20 0.48
KMT2A Q03164 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
MEN1 O00255 1/20 0.48
CYP3A4 P08684 1/20 0.47
GAA P10253 1/20 0.47
CYP2C9 P11712 1/20 0.47
ACP1 P24666 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474248 0.81 PSMB8 (0.57) CA1CA2CA12CA4CA7
SCHEMBL6985918 0.80 SMN1; SMN2 (0.58) CA1CA2CA12CA4CA7
SCHEMBL8799206 0.80 CA1 (0.54) CA1CA2CA12CA4CA7
SCHEMBL8799542 0.78 CA1 (0.55) CA1CA2CA12CA4CA7
SCHEMBL8229512 0.77 PSMB8 (0.64) CA1CA2CA12CA4CA7
SCHEMBL6976206 0.76 CA1 (0.50) CA1CA2CA12CA4CA7
SCHEMBL31452859 0.76 TARS1 (0.61) CA1CA2CA12CA4CA7
SCHEMBL3282188 0.74 PSMB8 (0.55) CA1CA2CA12CA4CA7
SCHEMBL10474769 0.74 PSMB8 (0.64) CA1CA2CA12CA4CA7
SCHEMBL9722824 0.74 CA1 (0.54) CA1CA2CA12CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355827-B1 Hydantoin derivatives MOCHIDA PHARM CO LTD (JP) 1997-01-02 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed