SCHEMBL8799744

SCHEMBL8799744

O=C1CN(S(=O)(=O)c2cc(-c3ccccc3)c(-c3ccccc3)s2)C(=O)N1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
PTP4A3 O75365 2/20 0.35
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
MAPK1 P28482 1/20 0.33
MMP2 P08253 1/20 0.32
KCNN4 O15554 1/20 0.32
KCNA3 P22001 1/20 0.32
PTP4A2 Q12974 1/20 0.32
PTP4A1 Q93096 1/20 0.32
PKM P14618 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HSD17B1 P14061 1/20 0.31
TDP2 O95551 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799405 0.89 POLB (0.37) POLBALDH1A1MAPTPTP4A3HSD17B10
SCHEMBL5953051 0.75 CA2 (0.49) POLBALDH1A1MAPTHSD17B10MEN1
SCHEMBL8972689 0.71 ALDH1A1 (0.69) POLBALDH1A1MAPTHSD17B10MEN1
SCHEMBL8799401 0.70 POLB (0.44) POLBALDH1A1MAPTHSD17B10MEN1
SCHEMBL8798618 0.70 HSD17B1 (0.39) ALDH1A1PTP4A3HSD17B10TDP1HSD17B1
SCHEMBL8799201 0.68 HDAC3 (0.37) POLBALDH1A1MAPTHSD17B10MEN1
SCHEMBL8799786 0.68 HDAC3 (0.37) POLBALDH1A1MAPTHSD17B10MEN1
SCHEMBL8797869 0.67 POLB (0.43) POLBALDH1A1MAPTMEN1KMT2A
SCHEMBL8799290 0.67 F10 (0.47)
SCHEMBL8798949 0.67 CA2 (0.34) POLBALDH1A1MAPTMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355827-B1 Hydantoin derivatives MOCHIDA PHARM CO LTD (JP) 1997-01-02 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed