SCHEMBL8799888

SCHEMBL8799888

Nc1nccc(C(=O)c2ccccc2OC(F)(F)F)c1C(=O)Cl

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.43
HCRTR1 O43613 7/20 0.38
HCRTR2 O43614 7/20 0.38
KCNK3 O14649 3/20 0.36
KCNK9 Q9NPC2 3/20 0.36
ATR Q13535 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
MGLL Q99685 1/20 0.34
ANO1 Q5XXA6 1/20 0.34
ELANE P08246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7542152 0.89 CDK2 (0.44) CDK2HCRTR1HCRTR2KCNK3KCNK9
SCHEMBL8798631 0.84 RORB (0.47) CDK2HSD17B10
SCHEMBL8610774 0.81 CNR2 (0.49) CDK2HTTHSD17B10
SCHEMBL7552945 0.79 ALDH1A1 (0.49) CDK2HTT
SCHEMBL8800986 0.78 RECQL (0.48) CDK2
SCHEMBL8799820 0.77 ALDH1A1 (0.40) HSD17B10ELANE
SCHEMBL7548471 0.77 MAPK13 (0.41) CDK2ELANE
SCHEMBL20641943 0.77 SCN9A (0.40) CDK2HCRTR1HCRTR2KCNK3KCNK9
SCHEMBL5784212 0.77 ELANE (0.52) CDK2HCRTR1HCRTR2KCNK3KCNK9
SCHEMBL7543771 0.74 BCAT2 (0.44) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-A1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-12-10 EP disclosed