SCHEMBL8799963

SCHEMBL8799963

O=C(O)N(CCCl)c1ccc(CC(F)(F)F)c([N+](=O)[O-])c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
MAPT P10636 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
GSTO1 P78417 1/20 0.35
ALDH1A1 P00352 5/20 0.34
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
PDK1 Q15118 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
AR P10275 1/20 0.31
PTGS2 P35354 1/20 0.31
CYP19A1 P11511 1/20 0.31
LMNA P02545 2/20 0.31
HPD P32754 1/20 0.31
HCAR3 P49019 1/20 0.30
ACLY P53396 1/20 0.30
GMNN O75496 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799973 1.00 CYP1A2 (0.39) CYP1A2MAPTNPC1RAB9AGSTO1
SCHEMBL16701743 0.79 TDP1 (0.44) CYP1A2MAPTNPC1RAB9AGSTO1
SCHEMBL8618765 0.76 SMN1; SMN2 (0.50) MAPTNPC1RAB9AALDH1A1TSHR
SCHEMBL8952221 0.76 SMN1; SMN2 (0.50) MAPTNPC1RAB9AALDH1A1TSHR
SCHEMBL27688694 0.72 CASP6 (0.58) TSHRPDK1LMNAHCAR3
SCHEMBL25245525 0.70 MAPK1 (0.49) CYP1A2MAPTALDH1A1TSHRTDP1
SCHEMBL27722916 0.69 TDP1 (0.50) CYP1A2MAPTRAB9AALDH1A1TSHR
SCHEMBL12090353 0.68 TSHR (0.55) CYP1A2MAPTNPC1RAB9AALDH1A1
SCHEMBL27856589 0.68 S100A4 (0.42) CYP1A2RAB9AALDH1A1TSHRTDP1
SCHEMBL8799965 0.68 ALDH1A1 (0.46) CYP1A2MAPTNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532039-B1 N1-trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes BRISTOL MYERS SQUIBB CO (US) 1997-12-03 EP disclosed
US-5260488-A Hair dye CLAIROL INC. (US) 1993-11-09 US disclosed
EP-0532039-A1 N1-trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes Bristol-Myers Squibb Company (US) 1993-03-17 EP disclosed
US-5186716-A N1 trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes and hair dyeing compositions and methods thereof CLAIROL INCORPORATED (US) 1993-02-16 US disclosed