SCHEMBL8800318

SCHEMBL8800318

COC(=O)[C@H](CCC(N)=O)NC(=O)CC1OC1C(Cc1ccccc1)NC(=O)[C@@H](CC(N)=O)NC(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.52
CTSB P07858 1/20 0.52
BACE1 P56817 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.43
MME P08473 2/20 0.43
ECE1 P42892 2/20 0.43
REN P00797 1/20 0.42
CAPN1 P07384 1/20 0.42
CTSL P07711 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801460 0.94 CTSD (0.52) CTSDCTSBSMN1; SMN2MMEECE1
SCHEMBL9412784 0.88 CTSD (0.52) CTSDCTSBRENCTSL
SCHEMBL8801156 0.84 CTSD (0.77) CTSDREN
SCHEMBL7298678 0.84 MME (0.53) CTSBSMN1; SMN2MMEECE1CTSL
SCHEMBL7295499 0.84 CTSL (0.51) CTSDCTSBMMEECE1CTSL
SCHEMBL9190618 0.83 CTSD (0.54) CTSDCTSBMMEECE1REN
SCHEMBL8664364 0.82 CTSD (0.49) CTSDCTSBCAPN1CTSLADORA3
SCHEMBL8661021 0.81 SMN1; SMN2 (0.48) CTSBSMN1; SMN2MMEECE1CTSL
SCHEMBL8663687 0.81 CTSD (0.47) CTSDCTSBMMEECE1CTSL
SCHEMBL8944865 0.79 CTSL (0.50) CTSDCTSBMMEECE1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP claimed