SCHEMBL8944865

SCHEMBL8944865

NC(=O)C[C@@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C1OC1CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 9/20 0.50
TACR1 P25103 2/20 0.47
CTSB P07858 3/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
MME P08473 1/20 0.46
ECE1 P42892 1/20 0.46
CTSD P07339 1/20 0.46
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8663687 0.97 CTSD (0.47) CTSLTACR1CTSBCTSSCTSK
SCHEMBL8944981 0.92 CTSD (0.48) CTSLCTSBCTSKMMEECE1
SCHEMBL7295499 0.89 CTSL (0.51) CTSLTACR1CTSBCTSSCTSK
SCHEMBL8661021 0.88 SMN1; SMN2 (0.48) CTSLCTSBMMEECE1
SCHEMBL8662047 0.88 PSMB1 (0.54) CTSLCTSBCTSSCTSK
SCHEMBL8664364 0.88 CTSD (0.49) CTSLCTSBCTSKCTSD
SCHEMBL8660791 0.84 CTRB1 (0.50) CTSLTACR1CTSBCTSSCTSK
SCHEMBL8665786 0.81 CTSD (0.48) CTSLCTSDKDM1A
SCHEMBL8944978 0.81 CTSS (0.56) CTSLCTSBCTSSCTSD
SCHEMBL8669118 0.81 CTSD (0.49) CTSLCTSBCTSSCTSKMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587388-A AIDS; VIRICIDES LUCKY LIMITED (KR) 1996-12-24 US disclosed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP disclosed