SCHEMBL7086183

SCHEMBL7086183

CC(=O)OC(C)c1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SLC6A9 P48067 2/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
ALDH1A1 P00352 3/20 0.34
PPP1CA P62136 1/20 0.34
KMT2A Q03164 1/20 0.34
GRM5 P41594 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
RXFP1 Q9HBX9 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
AGTR1 P30556 1/20 0.33
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800407 0.93 MEN1 (0.33) TP53ALDH1A1KMT2ASMN1; SMN2AGTR1
SCHEMBL8800780 0.90 PTGDR2 (0.35) TP53ALDH1A1KMT2ASMN1; SMN2NPSR1
SCHEMBL8799402 0.90 S1PR3 (0.37) SLC6A9GRIN1GRIN2BALDH1A1KMT2A
SCHEMBL8801551 0.87 TDP1 (0.36) TP53SLC6A9ALDH1A1KMT2ARXFP1
SCHEMBL8800655 0.87 CFTR (0.41) MAPTNPC1RAB9AALDH1A1KMT2A
SCHEMBL7081438 0.86 TP53 (0.36) TP53MAPTNPC1RAB9ASLC6A9
SCHEMBL6961698 0.86 S1PR3 (0.38) ALDH1A1KDM4E
SCHEMBL8802789 0.85 TP53 (0.37) TP53MAPTNPC1RAB9ASLC6A9
SCHEMBL7081153 0.84 MAPT (0.39) TP53MAPTNPC1RAB9ASLC6A9
SCHEMBL8801745 0.84 ALDH1A1 (0.40) TP53NPC1GRIN1GRIN2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed