SCHEMBL6967425

SCHEMBL6967425

CC(=O)OCc1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 2/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRM5 P41594 1/20 0.35
GABRA5 P31644 3/20 0.34
GABRA1 P14867 2/20 0.34
NPC1 O15118 2/20 0.34
SLC16A3 O15427 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
P2RX7 Q99572 1/20 0.34
PKM P14618 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
KMT2A Q03164 1/20 0.34
S1PR3 Q99500 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973275 0.93 ALDH1A1 (0.36) ALDH1A1TP53GABRA5GABRA1SLC16A3
SCHEMBL7084645 0.93 ALDH1A1 (0.38) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL6967707 0.92 ALDH1A1 (0.40) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL7086211 0.92 ALDH1A1 (0.39) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL7081541 0.91 IDO1 (0.35) TP53TDP1KMT2A
SCHEMBL7078901 0.91 ALDH1A1 (0.40) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL6972338 0.90 GRIN1 (0.38) ALDH1A1LMNAGRIN1GRIN2BPKM
SCHEMBL6969306 0.89 KMT2A (0.39) ALDH1A1LMNAGABRA5GABRA1TDP1
SCHEMBL6972994 0.88 RXFP1 (0.41) ALDH1A1LMNAKMT2A
SCHEMBL7085898 0.88 ALDH1A1 (0.37) ALDH1A1LMNATP53GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed