SCHEMBL8801798

SCHEMBL8801798

COc1cc(N)c(Cl)cc1C(=O)OCC1CCCCN1C

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 4/20 0.64
ACHE P22303 1/20 0.64
CYP3A4 P08684 2/20 0.64
GLA P06280 1/20 0.64
MEN1 O00255 1/20 0.61
ALDH1A1 P00352 1/20 0.61
CYP2D6 P10635 1/20 0.61
HTR3A P46098 1/20 0.61
KMT2A Q03164 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803953 0.83 HTR4 (0.60) HTR4ACHEALDH1A1
SCHEMBL9117844 0.81 HTR4 (0.70) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL17709629 0.78 ACHE (1.00) HTR4ACHECYP3A4GLA
SCHEMBL8803576 0.78 HTR4 (0.54) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL2579561 0.78 HTR4 (1.00) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL29386039 0.78 HTR4 (1.00) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL6774093 0.77 CHRNB4 (0.50) HTR4ACHECYP3A4GLA
Hydrochloric Acid SCHEMBL22532550 0.77 HTR4 (0.98) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL29767008 0.76 HTR4 (1.00) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL548053 0.76 HTR4 (1.00) HTR4CYP3A4GLAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0499995-B1 Piperidine derivatives NISSHIN FLOUR MILLING CO (JP) 1997-01-02 EP disclosed
US-5246945-A 5-hydroxytryptamine antagonist for nervous system disorders NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-09-21 US disclosed
EP-0499995-A2 Piperidine derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-08-26 EP disclosed