SCHEMBL8803576

SCHEMBL8803576

COc1cc(N)c(Cl)cc1C(=O)OC(C)C1CCCCN1C

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 4/20 0.54
CYP3A4 P08684 2/20 0.54
GLA P06280 1/20 0.54
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP2D6 P10635 1/20 0.53
HTR3A P46098 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8802995 0.83 HTR4 (0.47) HTR4ALDH1A1
SCHEMBL8801798 0.78 HTR4 (0.64) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL8801807 0.78 GAA (0.52) HTR4
SCHEMBL8295294 0.74 HTR4 (0.47) HTR4HTR3A
Hydrochloric Acid SCHEMBL9345072 0.74 HTR4 (0.61) HTR4CYP3A4MEN1ALDH1A1CYP2D6
SCHEMBL8803626 0.73 GRM1 (0.42) ALDH1A1
SCHEMBL15652199 0.73 MEN1 (0.66) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL7202734 0.73 HTR4 (0.57) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL28749742 0.73 HTR4 (0.65) HTR4CYP3A4GLAMEN1ALDH1A1
SCHEMBL9117844 0.72 HTR4 (0.70) HTR4CYP3A4GLAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0499995-B1 Piperidine derivatives NISSHIN FLOUR MILLING CO (JP) 1997-01-02 EP disclosed
US-5246945-A 5-hydroxytryptamine antagonist for nervous system disorders NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-09-21 US disclosed
EP-0499995-A2 Piperidine derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-08-26 EP disclosed