SCHEMBL8802015

SCHEMBL8802015

CC(=O)N[C@@H](C)C(=O)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.46
MTNR1B P49286 6/20 0.46
PGR P06401 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
HTR2A P28223 1/20 0.46
HRH1 P35367 1/20 0.46
KCNH2 Q12809 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
LMNA P02545 2/20 0.44
CTRC Q99895 1/20 0.44
ACACB O00763 1/20 0.43
ACACA Q13085 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10523295 1.00 MTNR1A (0.46) MTNR1AMTNR1BPGRADRA2AADRA2B
SCHEMBL1287117 0.86 PGR (0.47) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL3495542 0.86 PGR (0.47) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL5700509 0.84 SMN1; SMN2 (0.54) KMT2AALDH1A1LMNA
SCHEMBL11776569 0.82 KMT2A (0.47) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL6490420 0.82 PGR (0.44) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL28550392 0.82 L3MBTL1 (0.48) MTNR1AMTNR1BTDP1L3MBTL1ALDH1A1
SCHEMBL10949351 0.81 TSHR (0.48) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL19323907 0.81 KMT2A (0.48) MTNR1AMTNR1BPGRADRA2AADRA2B
SCHEMBL19323897 0.81 KMT2A (0.48) MTNR1AMTNR1BPGRADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0754041-A4 NOVEL SUBSTITUTED TRYPTAMINES, PHENALKYLAMINES AND RELATED COMPOUNDS INTERNEURON PHARMA (US) 1997-11-19 EP claimed
EP-0754041-A1 NOVEL SUBSTITUTED TRYPTAMINES, PHENALKYLAMINES AND RELATED COMPOUNDS INTERNEURON PHARMACEUTICALS INCORPORATED (US) 1997-01-22 EP claimed
US-4277420-A Ephedrine and pseudoephedrine precursors MONSANTO COMPANY (US) 1981-07-07 US disclosed