SCHEMBL8802020

SCHEMBL8802020

O=C(O)c1cn(-c2ccc(Cn3ccnn3)cc2)c2c(Cl)c(N3CCN(c4ccccc4Cl)CC3)c(F)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 3/20 0.42
POLB P06746 2/20 0.42
HSP90AA1 P07900 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TOP2A P11388 5/20 0.40
TOP2B Q02880 4/20 0.40
TOP1 P11387 3/20 0.40
PIM1 P11309 1/20 0.40
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8802022 0.91 CYP3A4 (0.35) CYP3A4CYP2C9KDM4EALDH1A1POLB
SCHEMBL8802764 0.90 CYP3A4 (0.45) CYP3A4CYP2C9KDM4EALDH1A1POLB
SCHEMBL8803805 0.88 KDM4E (0.45) CYP3A4CYP2C9KDM4EALDH1A1POLB
SCHEMBL8802244 0.87 KDM4E (0.42) CYP3A4CYP2C9KDM4EALDH1A1POLB
SCHEMBL8801501 0.86 HPGD (0.51) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL8801565 0.84 PIM1 (0.47) CYP3A4CYP2C9KDM4EALDH1A1POLB
SCHEMBL8801930 0.82 LMNA (0.57) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL8802774 0.81 CYP3A4 (0.36) CYP3A4CYP2C9KDM4EALDH1A1POLB
SCHEMBL8803902 0.80 ALDH1A1 (0.52) KDM4EALDH1A1POLBHSP90AA1RXFP1
SCHEMBL5522810 0.79 HPGD (0.49) CYP3A4CYP2C9KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612731-B1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1997-08-20 EP disclosed
EP-0612731-A1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1994-08-31 EP disclosed