SCHEMBL8801501

SCHEMBL8801501

O=C(O)c1cn(-c2ccc(Cn3ccnn3)cc2)c2c(F)c(N3CCN(c4ccccc4)CC3)c(F)cc2c1=O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.51
HSD17B10 Q99714 3/20 0.51
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 4/20 0.45
POLB P06746 1/20 0.45
HSP90AA1 P07900 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
TOP1 P11387 6/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41
TOP2A P11388 5/20 0.40
TOP2B Q02880 3/20 0.40
PIM1 P11309 2/20 0.40
ADRA2B P18089 1/20 0.39
MAPK1 P28482 1/20 0.39
PMP22 Q01453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801505 0.91 HPGD (0.42) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8802764 0.88 CYP3A4 (0.45) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8802020 0.86 CYP3A4 (0.43) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8803902 0.86 ALDH1A1 (0.52) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8801930 0.85 LMNA (0.57) HPGDHSD17B10KDM4EALDH1A1TOP1
SCHEMBL8803108 0.84 LMNA (0.44) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8801565 0.83 PIM1 (0.47) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8802774 0.81 CYP3A4 (0.36) HPGDHSD17B10KDM4EALDH1A1POLB
SCHEMBL8801262 0.80 LMNA (0.57) HPGDHSD17B10KDM4EALDH1A1TOP1
SCHEMBL8804229 0.80 LMNA (0.64) HPGDHSD17B10KDM4EALDH1A1TOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612731-B1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1997-08-20 EP disclosed
EP-0612731-A1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1994-08-31 EP disclosed