SCHEMBL8802995

SCHEMBL8802995

COc1cc(N)ccc1C(=O)OC(C)C1CCCCN1C

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 4/20 0.47
ACHE P22303 2/20 0.45
ALDH1A1 P00352 1/20 0.44
CASP6 P55212 1/20 0.41
CHRNB4 P30926 4/20 0.41
CHRNA3 P32297 4/20 0.41
CRBN Q96SW2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803576 0.83 HTR4 (0.54) HTR4ALDH1A1
SCHEMBL8803626 0.81 GRM1 (0.42) ACHEALDH1A1CHRNB4CHRNA3
SCHEMBL8803961 0.77 SLC6A3 (0.48) HTR4ACHEALDH1A1CASP6CRBN
SCHEMBL8803953 0.77 HTR4 (0.60) HTR4ACHEALDH1A1CHRNB4CHRNA3
SCHEMBL7154189 0.72 MEN1 (0.65) HTR4ACHEALDH1A1
SCHEMBL10156660 0.71 HPGD (0.67) HTR4ACHEALDH1A1
SCHEMBL7278288 0.70 HTR3E (0.56) HTR4ALDH1A1CHRNB4CHRNA3
SCHEMBL7271032 0.70 HTR3E (0.56) HTR4ALDH1A1CHRNB4CHRNA3
SCHEMBL5925494 0.69 GAA (0.64) ALDH1A1CRBN
SCHEMBL13880742 0.69 CRBN (0.57) HTR4ACHEALDH1A1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0499995-B1 Piperidine derivatives NISSHIN FLOUR MILLING CO (JP) 1997-01-02 EP disclosed
US-5246945-A 5-hydroxytryptamine antagonist for nervous system disorders NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-09-21 US disclosed
EP-0499995-A2 Piperidine derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-08-26 EP disclosed