SCHEMBL8804735

SCHEMBL8804735

NS(=O)(=O)c1ccc(NC(=O)c2cccnc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.77
CYP3A4 P08684 2/20 0.74
CYP2C9 P11712 1/20 0.74
ALDH1A1 P00352 4/20 0.70
CA1 P00915 2/20 0.68
CA2 P00918 2/20 0.68
CA12 O43570 1/20 0.68
CA9 Q16790 1/20 0.68
KMT2A Q03164 2/20 0.67
POLB P06746 1/20 0.67
MEN1 O00255 1/20 0.67
ROCK2 O75116 1/20 0.66
ROCK1 Q13464 1/20 0.66
SMN1; SMN2 Q16637 3/20 0.64
GAA P10253 2/20 0.64
LMNA P02545 1/20 0.63
HIF1A Q16665 1/20 0.63
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
TP53 P04637 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14679077 0.85 CYP3A4 (1.00) L3MBTL1CYP3A4CYP2C9ALDH1A1KMT2A
SCHEMBL161057 0.84 CYP3A4 (0.81) CYP3A4CYP2C9ALDH1A1KMT2APOLB
SCHEMBL3518422 0.84 IKBKB (0.64) L3MBTL1POLB
SCHEMBL10327416 0.82 ALDH1A1 (0.80) CYP3A4CYP2C9ALDH1A1KMT2APOLB
SCHEMBL29596938 0.82 ALDH1A1 (1.00) L3MBTL1CYP3A4CYP2C9ALDH1A1KMT2A
SCHEMBL3093633 0.82 CYP3A4 (0.82) CYP3A4CYP2C9ALDH1A1KMT2AMEN1
SCHEMBL8422583 0.82 CA2 (1.00) CYP2C9CA1CA2CA12CA9
SCHEMBL15598889 0.81 CYP3A4 (0.74) L3MBTL1CYP3A4CYP2C9ALDH1A1KMT2A
SCHEMBL29596226 0.81 ROCK2 (0.71) CYP3A4CYP2C9ALDH1A1KMT2AMEN1
SCHEMBL3093627 0.81 ROCK2 (0.71) CYP3A4CYP2C9ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1155278-A Arylthio compounds as antibacteral and antiviral agents WARNER LAMBERT CO (US) 1997-07-23 CN claimed
EP-0775110-A1 ARYLTHIO COMPOUNDS AS ANTIBACTERIAL AND ANTIVIRAL AGENTS WARNER-LAMBERT COMPANY (US) 1997-05-28 EP claimed
WO-1996004242-A1 ARYLTHIO COMPOUNDS AS ANTIBACTERIAL AND ANTIVIRAL AGENTS WARNER-LAMBERT COMPANY (US) 1996-02-15 WO claimed