SCHEMBL8807141

SCHEMBL8807141

CCOC(=S)c1c[nH]c(C)n1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA9 Q16790 2/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801869 0.78 CYP1A2 (0.55) CYP1A2KMT2AMEN1
SCHEMBL441004 0.72
SCHEMBL20268120 0.70 ALDH1A1 (0.43) CYP1A2CA12CA1CA2CA9
SCHEMBL2852145 0.67 NOTUM (0.32)
SCHEMBL1040746 0.67 NOTUM (0.32)
SCHEMBL8887619 0.67 BAZ2B (0.50) CYP1A2KMT2ATDP1
SCHEMBL170375 0.66
SCHEMBL3861670 0.66
SCHEMBL1204641 0.66
SCHEMBL8808976 0.66 LPO (0.38) CYP1A2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785937-A1 2-(IMIDAZOL-4-YL)CARBAPENEME DERIVATIVES, INTERMEDIATES THEREOF AND USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1997-07-30 EP disclosed
WO-1996011932-A1 2-(IMIDAZOL-4-YL)CARBAPENEME DERIVATIVES, INTERMEDIATES THEREOF AND USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1996-04-25 WO disclosed