SCHEMBL8809208

SCHEMBL8809208

CC(=O)Oc1cccc(Oc2cc(OCc3ccccc3)ccc2C#N)c1C

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.51
MRGPRX4 Q96LA9 2/20 0.51
PTPN1 P18031 1/20 0.46
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809211 0.85 MAOB (0.54) MAOBMRGPRX4PTPN1
SCHEMBL8814943 0.83 AR (0.37) MAOBMRGPRX4
SCHEMBL12988735 0.83 MAOB (0.70) MAOBMRGPRX4PTPN1
SCHEMBL8808914 0.77 MRGPRX4 (0.45) MAOBMRGPRX4
SCHEMBL8896538 0.76 PTPN1 (0.63) MAOBMRGPRX4PTPN1
SCHEMBL8808917 0.76 XDH (0.45) MAOBMRGPRX4
SCHEMBL8133729 0.75 CYP19A1 (0.47) MAOBMRGPRX4
SCHEMBL3865512 0.75 MAOB (0.77) MAOBMRGPRX4
SCHEMBL7404465 0.75 MAOB (0.63) MAOBMRGPRX4
SCHEMBL6199191 0.75 PTPN1 (0.59) MAOBPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805802-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE-POULENC RORER LIMITED (GB) 1997-11-12 EP disclosed
WO-1996022978-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LIMITED (GB) 1996-08-01 WO disclosed