SCHEMBL8809394

SCHEMBL8809394

O=C1CC(Oc2ccccc2OCc2ccccc2)N1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 3/20 0.54
BRD4 O60885 3/20 0.54
TNKS2 Q9H2K2 2/20 0.46
SLC6A4 P31645 4/20 0.44
HTR1A P08908 3/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A3 Q01959 2/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TTR P02766 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4059320 0.77 CREBBP (0.45) CREBBPBRD4MAPTALDH1A1HTT
SCHEMBL9559115 0.74 CREBBP (0.43) CREBBPBRD4PDE4APDE4BPDE4C
SCHEMBL339812 0.74 MAPT (0.71) BRD4HTR1ASLC6A2SLC6A3MAPT
SCHEMBL27767020 0.73 MAOB (0.56) CREBBPBRD4TNKS2SLC6A2SLC6A3
SCHEMBL5207455 0.73 MAOB (0.56) CREBBPBRD4TNKS2SLC6A2SLC6A3
Formaldehyde SCHEMBL27831678 0.72 MAPT (0.63) BRD4HTR1AMAPTMAPK1TDP1
SCHEMBL7360048 0.71 ALOX5 (0.50) CREBBPBRD4SLC6A4SLC6A2SLC6A3
SCHEMBL17680774 0.71 CREBBP (1.00) CREBBPBRD4
SCHEMBL10702878 0.70 BRD4 (0.47) CREBBPBRD4SLC6A2SLC6A3MAPK1
SCHEMBL23258867 0.69 MAPT (0.59) BRD4HTR1AMAPTMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO disclosed