SCHEMBL8819835

SCHEMBL8819835

O=C(O)CC1CCC=CC=N1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.33
GABRR1 P24046 4/20 0.33
GABRA5 P31644 4/20 0.33
GABRB2 P47870 4/20 0.33
GABRA4 P48169 4/20 0.33
SLC6A12 P48065 2/20 0.33
SLC6A13 Q9NSD5 2/20 0.33
SLC6A1 P30531 1/20 0.31
SLC6A11 P48066 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5140299 0.81 GABRA1 (0.34) GABRA1GABRR1GABRA5GABRB2GABRA4
SCHEMBL7854558 0.71 SLC6A12 (0.35) GABRA1GABRR1GABRA5GABRB2GABRA4
SCHEMBL7072429 0.65 SLC6A12 (0.45) GABRA1GABRR1GABRA5GABRB2GABRA4
SCHEMBL459030 0.61
SCHEMBL971678 0.61
SCHEMBL10296559 0.60
SCHEMBL92858 0.60 KDM4E (0.43) GABRA1GABRR1GABRA5GABRB2GABRA4
SCHEMBL22587458 0.60 KDM4E (0.43) GABRA1GABRR1GABRA5GABRB2GABRA4
Hydrochloric Acid SCHEMBL10808909 0.60 CHRNB2 (0.49) GABRA1GABRR1GABRA5GABRB2GABRA4
SCHEMBL11579290 0.59 TSHR (0.46) GABRA1GABRA5GABRB2GABRA4SLC6A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997047624-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed
WO-1997047625-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed