SCHEMBL8828210

SCHEMBL8828210

O=C(O)C/C=C/c1ccc2c(c1)OCO2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.60
CYP1A2 P05177 1/20 0.60
HDAC6 Q9UBN7 2/20 0.55
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 3/20 0.55
TRPM8 Q7Z2W7 2/20 0.55
GAA P10253 1/20 0.54
CYP3A4 P08684 2/20 0.54
ATM Q13315 1/20 0.54
TDP1 Q9NUW8 1/20 0.53
MAOB P27338 1/20 0.52
CYP19A1 P11511 1/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
MTOR P42345 1/20 0.51
VCP P55072 1/20 0.51
CYP2D6 P10635 1/20 0.51
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828230 1.00 HSD17B10 (0.60) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL20702283 0.82 ALDH1A1 (0.53) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL14552385 0.81 SOAT1 (0.56) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL2453908 0.80 CYP3A4 (0.61) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL2005021 0.80 CYP3A4 (0.61) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL15517799 0.79 MAOA (0.60) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL15509220 0.79 MAOA (0.60) HSD17B10CYP1A2HDAC6HDAC3HDAC1
SCHEMBL4745288 0.79 KDM4E (0.81) HSD17B10CYP1A2HDAC6ALDH1A1KDM4E
SCHEMBL79427 0.79 KDM4E (0.81) HSD17B10CYP1A2HDAC6ALDH1A1KDM4E
SCHEMBL1254171 0.79 ALDH1A1 (0.62) HSD17B10CYP1A2HDAC6HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed