SCHEMBL8828231

SCHEMBL8828231

COc1ccc(CCN(C)CCCNC(=O)C/C=C/c2cccc(-n3ccnc3)c2)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.44
TMEM97 Q5BJF2 3/20 0.44
SIGMAR1 Q99720 3/20 0.44
HPGD P15428 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
NOS2 P35228 2/20 0.40
CYP3A4 P08684 2/20 0.40
QPCT Q16769 1/20 0.40
PKM P14618 2/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 2/20 0.39
OPRK1 P41145 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
SMPD1 P17405 3/20 0.39
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828195 0.92 OPRM1 (0.44) OPRM1TMEM97SIGMAR1HPGDNOS2
SCHEMBL9233122 0.89 OPRM1 (0.42) OPRM1TMEM97SIGMAR1HPGDNOS2
SCHEMBL8828256 0.87 OPRM1 (0.43) OPRM1TMEM97SIGMAR1HPGDNOS2
SCHEMBL9156928 0.84 OPRM1 (0.41) OPRM1TMEM97SIGMAR1HPGDNOS2
SCHEMBL8828422 0.84 OPRM1 (0.43) OPRM1TMEM97SIGMAR1HPGDNOS2
SCHEMBL8828362 0.84 LMNA (0.59) OPRM1TMEM97SIGMAR1HPGDLMNA
SCHEMBL8828168 0.84 DRD3 (0.45) SIGMAR1DRD2DRD3
SCHEMBL8828419 0.84 MAOB (0.38) OPRM1TMEM97SIGMAR1HTTPKM
SCHEMBL9160192 0.84 CYP3A4 (0.38) OPRM1TMEM97SIGMAR1HPGDCYP3A4
SCHEMBL9160628 0.83 MAOB (0.38) OPRM1TMEM97SIGMAR1NOS2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed