SCHEMBL8828232

SCHEMBL8828232

COc1ccc(CCN(C)CCCN(C)C(=O)C/C=C/c2ccc(-n3ccnc3)cc2)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
CYP3A4 P08684 5/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
SMPD1 P17405 5/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAOB P27338 1/20 0.41
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.40
HCN4 Q9Y3Q4 1/20 0.39
CDK8 P49336 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828359 0.88 KMT2A (0.39) ALDH1A1CYP3A4CYP1A2CYP2D6BLM
SCHEMBL8828195 0.87 OPRM1 (0.44) ALDH1A1CYP3A4CYP1A2CYP2D6BLM
SCHEMBL9233122 0.87 OPRM1 (0.42) ALDH1A1CYP3A4CYP1A2CYP2D6BLM
SCHEMBL8828347 0.83 POLB (0.40) ALDH1A1CYP3A4CYP1A2CYP2D6BLM
SCHEMBL8828234 0.83 CYP3A4 (0.50) ALDH1A1LMNACYP3A4CYP1A2CYP2D6
SCHEMBL9160192 0.81 CYP3A4 (0.38) ALDH1A1CYP3A4KDM4ESMN1; SMN2MAOB
SCHEMBL8828270 0.81 ALDH1A1 (0.39) ALDH1A1CYP3A4CYP1A2CYP2D6KDM4E
SCHEMBL9160628 0.80 MAOB (0.38) MAOB
SCHEMBL8828417 0.80 L3MBTL1 (0.42) ALDH1A1LMNACYP3A4KDM4ESMN1; SMN2
SCHEMBL8828419 0.79 MAOB (0.38) ALDH1A1KDM4EMAOBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed